Lomitapide可經由抑制三酸甘油酯和膽固醇轉化為極低密度脂蛋白(VLDL),抑制乳糜微粒合成,達到降低血漿中低密度膽固醇(LDL-C)的濃度,其藥理作用機制為何?
Apo B inhibitor
mitochondrial transition pore inhibitor
proprotein convertase subtilisin/kexin type 9 inhibitor
microsomal triglyceride transfer protein inhibitor